Ex parte OIDA et al. - Page 14




               Appeal No. 94-4265                                                                                                      
               Application 08/035,915                                                                                                  






                                         10                                                        11                             
                               wherein R  represents a hydrogen atom or a C -C  alkyl group and R  represents a                        
                                                                                1   4                                                  
                               hydrogen atom, allyloxycarbonyl, 2-methylallyloxycarbonyl, 2-chloroallyloxy-                            
                               carbonyl, 2,2,2-trichloroethoxy-carbonyl,  2,2,2-tribromoethoxycarbonyl,  p-nitro-                      
                               benzyloxycarbonyl or o-nitrobenzyloxycarbonyl,                                                          
               groups of the formula                                                                                                   






                                          12       13                                                                                  
                               wherein R  and R  are the same or different and each represents a hydrogen atom                         
                               or a C -C  alkyl group and Y represents an oxygen atom, a sulphur atom or an imino                      
                                      1  4                                                                                             
                               group which may be optionally substituted with a C -C  alkyl group,                                     
                                                                                     1   4                                             
               C -C  alkoxycarbonyl groups, benzyloxycarbonyl, phenethyloxycarbonyl, p-nitrobenzyloxycarbonyl                          
                 2  7                                                                                                                  
               and o-nitrobenzyloxy carbonyl group; and                                                                                
                               the substituents attached to the nitrogen atoms of the non-aromatic heterocyclic                        
                               groups may be substituted with one or more groups selected from the group                               
                               consisting of C -C  alkyl groups, C -C  alkoxy groups hydroxy, amino, halogen, C -1   4               1  4                ,                            1                 
                               C  aliphatic acyloxy groups, C -C  aliphatic acylarnino groups, cyano, azido, carboxy,1                                                                                        
                                 5                           1   5                                                                     
                               C -C  alkoxycarbonyl groups, the carbamoyl group, C -C  alkylthio group, C -C1                                                                         
                                 2   5                                                   1  4                    l  4                
                               alkylsulphinyl groups, C -C  alkylsulphonyl groups, nitro group, and groups of                          
                                                          1  4                                                                         
                               formula                                                                                                 






                                          14       15                                                                                  
                               wherein R  and R  are the same or different and each represents a hydrogen atom                         
                               or a C -C  alkyl group;                                                                                 
                                      1  4                                                                                             
                       a substituted alkyl group, said substituted alkyl groups being selected from the group consist-                 
               ing of a hydroxyalkyl group, a protected hydroxy alkyl group, an aminoalkyl group, and a protected                      
                                                                 -14-                                                                  





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